Genvoya waa hal kiniin ah, daroogo isku dhafan oo loo isticmaalo daaweynta HIV, kaas oo ka kooban afar daroogo oo daawada antiretroviral ah :
- Elvitegravir , isdhexgaliye isdhexgalka
- Cobicistat , daroogada HIV "daroogo"
- Emtricitabine, oo ah nucleotide celinta transcriptase inhibitor (NtRTI)
- Tenofovir alafenamide (TAF), NtRTI kale
Genvoya waa kiniinka isku dhafka ah ee ugu horreeya ee lagu isticmaalo TAF, oo ah "kobcin" oo ah "tayada" oo lagu magacaabo Tenofovir disoproxil fumarate (TDF) oo laga helo daawooyinka Truvada, Atripla , iyo Complera.
Sidan oo kale, waxaa loo tixgelin karaa horumarinta Stribild , hal-abuurka kiniinada oo ka kooban elvitegravir + cobicistat + emtricitabine + TDF.
TAF waxaa loo tixgeliyaa inay ka sarreyso TDF maadaama ay awood u leedahay in ay daawada ugu firfircoon si wax ku ool ah u isticmaasho unugyada iyo qiyaaso aad u yar-macnaheedu waxa weeye in aysan jirin wax yar ee daroogada ee ku jira dhiigga iyo in yar ka yaryihiin sidii loo kobcin lahaa kelyaha la xidhiidha daroogada sunta.
(Inkasta oo halista TDF-ku xirxirto sunta sunta ay tahay mid aad u hooseeya dalalka horumaray, khatartaas waxaa loo arkaa in ay si weyn u kicinayso dalalka soo koraya halkaasoo ay jirto xaalad weyn oo ka timaadda cillad kelyo horay u jirtay.
Calaamadaha daaweynta
Genvoya waxaa ansixiyay Maamulka Cuntada iyo Maandooriyeyaasha Mareykanka bishii November 5, 2015, iyaga oo isticmaala labadaba dadka waaweyn iyo caruurta da'doodu ka weyn tahay 12 sano oo aan waligood ku jirin daaweyn HIV iyo miisaankeedu yahay 77 rodol (35 kg). Waxaa sidoo kale loo oggol yahay dadka qaangaarka ah ee ku jira daaweynta kuwaas oo si buuxda u xakameynaya (aan la garan karin) fayruska .
Dejinta
Genvoya waa kiniin cagaaran, qallafsan, oo kiniin ah, oo ka kooban 150mg of elvitegravir, 150mg of cobicistat, 200mg of emtricitabine iyo 10mg of TAF. Waxaa lagu qoslaa "GSI" hal dhinac iyo "510" dhinaca kale.
Qiyaasta
Hal kiniin ayaa maalin walba la qaataa cunto. Genvoya waa in aan lagu qaadin dawooyinka kale ee daawooyinka antiretroviral ee loo isticmaalo daaweynta HIV.
Waxyaabaha kale ee saameynaya
Qaar ka mid ah saamaynta daroogada ayaa lagu qoray bukaanka bukaan socodka daaweynta qaadashada Genvoya. Dhacdooyinka ugu caansan ee lagu arko, oo lagu soo warramey 5% ama in ka badan oo bukaan ah, waa:
- Lalabbo
- Shuban
- Daal
- Madax xanuun
Dhibaatooyinka kale waxay ahaayeen kuwo caadi ah, oo xaliya muddada udhigma 1-2 toddobaad, iyadoo tiro yar oo ka mid ah bukaanada joojinayaan sababtoo ah dulqaadasho daaweyneed.
Khilaafaadka
Genvoya waa in aan la qaadin daroogooyinka soo socda ama dheeraadka ah:
Daawooyinka ka hortagga migreebka: Cafergot, Migergot, Ergostat, Dhexdhexaadiye Ergotamiin, Wigren, Wigreles, Ergotrate, Methergine, DHE 45
- Daawada anti-psikotikada: Orap
- Daawooyinka loo yaqaan "Statolitos": Zocor, Simcor, Vytorin, Mevacor, Advicor, Altoprev, Mevacor
- Dawada cagaarshowga B: Hepsera, Preveon
- Wakiilada Daawada: Daacad, Quicksolv Propulsid
- Daawooyinka Prostate: Uroxatral
- Daawooyinka dhiig-yari ee soodhoweyn: Revatio
- Dawooyinka ka hortaga qaaxada: Mycobutin, Rifater, Rifamate, Rimactane, Rifadin, Priftin
- Sedatives: Calaamadaha, Halcion
- St. John Wort
Tixgelinno Kale
Genvoya laguma talineynin bukaanka qaba naafanimada kalyaha (oo lagu qeexay inay tahay in la qiyaaso nadiifinta wax soo saarka ee wax ka yar 30mL daqiiqadii). Fadlan kugula tali dhakhtarkaaga haddii laguu daaweeyay ama lagu daaweynayo kalyo kasta ee dhakhtarka kale.
Genvoya laguma talineynin bukaanka qaba ciladda beerka ama kuwa qaba infakshanka cagaarshow B (HBV) ee daba dheeraaday sababta oo ah waxay si weyn u sii xumeyn kartaa dhibaatooyinka beerka. Waxaa lagula talinayaa in dadka qaba HIV lagu baaro HBV ka hor inta aysan qorin Genvoya. Fadlan kugula talinay dhakhtarkaaga haddii aad qabtid dhibaatooyin beerka iyo / ama taariikhda cagaarshow.
Ilaha:
Maamulka Cuntada iyo Dawooyinka Mareykanka. "FDA waxay ogolaatay daaweyn cusub oo HIV ah." Silver Spring, Maryland; saxaafadeed la soo saarey November 5, 2015.
Gilead Sciences. "Genvoya - Macluumaad Dheeraad Ah." Foster City, California