Qeybinta
Evotaz (atazanavir + cobicistat) waa daroogo goosad ah oo la isku daro daawada antiretroviral ee loo isticmaalo daaweynta HIV . Labada qaybood ee daroogada ayaa si gooni ah loo iibiyaa sida Reyataz (atazanavir) iyo Tybost (cobicistat) .
Isku-dubaridaha hal-hal-abuurka ah ayaa u oggolaanaya fududaan, qiyaasta daaweynta maalinlaha ah, iyada oo qayb ka mid ah " cobicistat " ay si wax ku ool ah u "kor u qaadeyso" iyo joogtaynta faytoominta atazanavir ee jirka.
Evotaz waxaa ansixiyay Maamulka Cunnada iyo Mukhaadaraadka ee Maraykanka (FDA) bishii Janaayo 2015 ee loogu talagalay bukaanada qaan-gaarka ah ee cusub iyo khibradba leh ee qaba HIV-1.
Foomka
Kiniin la duubay oo kakooban, oo ka kooban 300mg atazanavir iyo 150mg cobicistat, waa midab casaan ah oo ku duuban lambarada "3641" hal dhinac.
Qiyaasta
Hal kiniin ayaa maalin walba la qaataa cunto. Evotaz looma isticmaali karo keligiis, lakiin waa in la qaataa iyadoo la raacayo hal ama in ka badan oo ah daroogo antiretroviral ah.
Tilmaamaha
Ka hor intaan la bilaabin, bukaanka waa in la baaraa si loo qiimeeyo qiyaasta loo yaqaan 'cynineine' oo lagu qiyaasay maaddaama Evotaz ay dhici karto in ay waxyeeleyso kalyaha (kelyaha), inta badan dadka bukaanka qaba cilladda kelyaha ee la yaqaan ama aan la ogaan karin. Marka lagu daro Viread (tenofovir ) -a daroogo oo keeni karta cilladda kelyaha ee qaar ka mid ah-waxaa lagu talinayaa in bukaanku la baadho qiyaasta nadiifinta, glucose kaadi, iyo borootiinka kaadida.
Waxaa sidoo kale lagu talinayaa in bukaanada daaweyn-khibrad leh, gaar ahaan kuwa ku faafa xanuunka HIV protease , la siiyo baaritaanka caabuqa hiddaha ka hor inta aan lagu qorin Evotaz.
Haddii baaritaanada unugyada aan la heli karin, Evotaz waa in laga fogaadaa cidkasta oo horay u soo gaadhay xanuunka HIV protease.
Saameynada Caadiga ah
Qaybta 3aad ee cilmi-baarista bani-aadamka ee bani'aadamnimada, tiro badan oo saameyn ku yeelan kara daroogooyinka ayaa la ogaaday marka la isticmaalayo Evotaz. Dhacdooyinka ugu caansan, ee lagu soo warramey 2% ama ka yar bukaanka dhowaan la daweeyey, waxay ahaayeen:
- Jaundice (maqaarka haragga iyo indhaha)
- Maaskaro (maqaarka indhaha)
- Finan
- Lalabbo
Dhibaatooyinka caanka ah ee aan caadiga ahayn waxaa ka mid ah daal, madax-xanuun, hurdo, matag iyo xanuunka caloosha oo sareeya. Dhismayaasha kelyaha ayaa sidoo kale lagu xusay bukaanjiifka markii Evotaz lagu soo dhaweeyay Viread (tenofovir), inkastoo kiisaska loo qaddariyay khafiifin aynaan keenin joojinta daaweynta.
Astaamaynta Daroogada
Evotaz waa in aan lagu qaadin daawooyinka soo socda ama daawooyinka dabiiciga ah:
- Daawada anti-anginal: Ranexa
- Daawooyinka isdaba joogga ah: Multaq
- Dawooyinka anti-cholesterol: Mevacor, Zocor
- Dawooyinka lidka ku ah daawooyinka: Uroxatral
- Dawooyinka anti-hypertension: Revatio
- Daawooyinka ka hortagga maskaxda: Latuda, Orap
- Dawooyinka Kansarka: Camptosar, Campto
- Ergot-ka kooban walxaha dheef-shiid kiimiko ah: DHE 45, Ergotrate, Hydergine, Migranal
- Dawooyinka anti-tuberculosis ku salaysan Rifampin: Mycobutin, Rifater, Rifamate, Rimactane, Rifadin, Priftin
- Sedatives: Dormicum, Halcion, Hypam, Hyponvel, Trilam, Aasaasay
- St. John Wort
Isdhex galka daawada Antiretroviral
Isticmaalka Tybost iyadoo la raacayo daroogooyinka daawooyinka antiretrovoviral ayaa laga yaabaa in ay keenaan lumitaanka saameynta daaweynta ee daroogada raacsan ama korodhka saameynta daawooyinka:
- Crixivan (indinavir) looma ogolaanayo in lala xiriiriyo Evotaz.
- Intelis (etravirine) waa in aan lagu xirin Evotaz.
- Sustiva (efavirenz) looma ogolaanayo in lala xiriiriyo Evotaz.
- Viramune (nevirapine) looma ogolaanayo in lala xiriiriyo Evotaz.
- Selzentry (maraviroc) qiyaasta waa in la isku hagaajiyaa ilaa 150mg maalintii laba jeer maalintii haddii ay la socdaan Evotaz.
Isdhexgalka kale ama Tixgelinnada kale
- U sheeg dhakhtarkaaga wixii xaalad ah ee kalyaha ama kalyaha ah ee laga yaabo in aad qabtid ka hor inta aanad bilaabin Evotaz.
- La socodsii dhakhtarkaaga wixii xaalad ah ee la ogaan karo ama laga shakiyay (beerka) oo laga yaabo inaad horey u soo qaadatay Evotaz, oo ay ku jiraan cagaarshow A, cagaarshow B ama cagaarshow C.
- Antacids oo leh aluminium ama magnesium hydroxide waxay ka hortagi kartaa Evotaz in si habboon loo nuugo. Haddii aad isticmaasho antidit-ka-ka-soo-jiidka (sida Rolaids, Tums, Caano Magnesia), waxaa la soo jeedinayaa in la qaato laba saacadood ka hor ama ka dib qiyaasta Evotaz.
- H 2- Argaggixisada ayaa loo isticmaalaa in lagu xakameeyo astaamaha caloosha (tusaale ahaan, Tagamet, Pepcid, Axid, Zantac) ayaa sidoo kale xakamayn kara nuugista Evotaz. Waxaa la soo jeediyay in la qaato Evotaz ama, si kale, 10 saacadood ka hor ama ka dib qiyaasta Evotaz.
- Tareenka difaacaha (sida, Losec, Prilosec, Prevacid, Nexium, Pariet) waxay sidoo kale ka hortagi kartaa nuugista Evotaz. Waxaa lagu talinayaa in la qaato 12 saacadood ka hor ama ka dib qiyaasta Evotaz.
- Daawada maqnaashaha aan habooneyn (Viagra, Levitra, Cialis) waa in loo isticmaalaa taxaddar sida Evotaz ay kor u qaadi karto heerarka waxyeelo xun, oo ay ku jiraan waxyeelo muuqda, isku-buuqsanaanta, iyo horjoogsiga (xannuuno xanuun, joogto ah). Waxaa lagu talinayaa in qiyaasta Viagra loo yareeyo in ka badan 25mg 48 saacadood; Qiyaasta Levitra waa la yaraynayaa in ka badan 2.5mg 72 saacadood; iyo qiyaasta Cialis waa la yaraynayaa in ka badan 10mg 72 saacadood.
- Xilliga uurka, Evotaz waa in aan la qorin inta lagu jiro muddada labaad ama saddexaad, haddii bukaanka uurka leh uu qaato H 2- daweeye antagonist ama Viread (tenofovir) maadaama ay dhici karto inuu halis u yahay kernicterus (xaalad naadir ah oo ku dhacda dhalaanka cusub cagaarsho daran).
Ilaha:
Bristol-Myers Squibb. "Evotaz (Atazanvir + cobicistat) - MACLUUMAAD KU QORAN MACLUUMAAD". New York, New York; heley Febraayo 3, 2015.