Methimazole, Carbimazole iyo Propylthiouracil / PTU
Marka qanjidhada thyroid noqdaan kuwo aan firfircoonayn - xaalad loo yaqaan hyperthyroidism - qanjirka ayaa keena hormoon tayroodh ah. Tani, waxay noqon kartaa, inay sababi karto calaamado kala duwan, oo ay ka mid yihiin garaaca wadnaha, dhiig karka, walaaca, hurdo la'aanta, miisaanka, miisaanka, shubanka, iyo calaamado badan oo ah calaamadaha shucaaca, iyo qanjidhada aan jirka lahayn.
Daaweyn muhiim ah oo loogu talagalay hyperthyroidism waa qayb ka mid ah daawooyinka rijeetada loo yaqaan daawada antithyroid. Daawooyinka Antidiotiga waxaa sidoo kale loo yaqaannaa thioamides. Waa daawooyin loo isticmaalo daweynta thyroid-ka-dillaaca - hyperthyroidism - oo ay ku jiraan marka qanjiradu ka buuxdo cudurada Graves ', boogaha sunta ah, ama sunta sunta ah.
Dawooyinka antidiolokiyo waxay ku shaqeeyaan xannibista awoodda qanjirka 'thyrox' si ay u soo saaraan laba xabbadood oo muhiim ah oo tayroodh ah thyroxine (T4) iyo triiodotyronine (T3).
Dawooyinka muhiimka ah ee antithyroid ee Maraykanka waxaa laga heli karaa methimazole iyo propylthiouracil (PTU). Ka baxsan Maraykanka, doorashadu waa methimazole, carbimazole, iyo PTU.
Methimazole
Methimazole-da daawada antidiotide-ga wuxuu ka hortagaa dheef-shiid kiimikaad isticmaalaya iodine - badanaa cuntada ama dheellitirka - si loo soo saaro hoormoonka tayroodh. Waa daawo caadi ahaan la qaato bukaanka maalintii.
Methimazole waxaa mararka qaar loogu yeeraa magaca thiamazole.
Daroogadan waxaa loo isticmaalaa adduunka oo dhan waana daawada ugu muhiimsan ee daawada antithyroid ee Maraykanka, halkaas oo laga heli karo magaca Tapazole.
Qaar ka mid ah shirkaduhu waxay sidoo kale bixiyaan nooc guud oo ah methimazole.
Carbimazole
Carbimazole waa daroogada, marka la maamulo, waxay u badashaa methimazole daroogada, sidaas darteedna waa mid aad u fiican oo ficil ah.
Nooca ugu caansan ee carbimazole waa Neomercazole.
Neomercazole waa magac calaamadeysan oo ah carbimazole waxaana soo saarey Amdipharm International (UK). Daroogada ayaa la ansixiyey 2004, waxaana lagu iibiyaa UK iyo Europe, laakiin lagama helayo ama lagu qorey Maraykanka. Waxaad ka arki kartaa macluumaadka ku yaal Neomercazole halkan. Waa kuwan dhowr waxyaalood oo dheeraad ah oo ku saabsan Neomercazole.
- Websaytka Maandooriyaha: Amdipharm
- Macluumaadka Qorista
Neomercazole Waxyaabaha : Carbimazole Ph.Eur; lactose; miraayada galleyda; sukrose; magnesium stearate; sukrose; talc; gum acacia; Dheriga Oxide; propyl hydroxybenzoate; iyo jelatin.
Xoogagga la heli karo : 5 mg
Noocyada / Magacyada kale: Carbimazole waxaa laga heli karaa qaar ka mid ah wadamada Yurubta iyo Aasiya sida ku cad magacyada calaamadaha soo socda: Atirozidina, Basolest, CG1, Carbimazole Spofa, Carbotiroid, Mertiran, Neo-Mercazole, Neo-Thierostat, Neo-Tireol, iyo Tyrazol.
Propylthiouracil / PTU
Habka PTU wuxuu hoos u dhigi karaa hormoonka tayroodhka hoormoonka tayroodh waa inuu joojiyaa qanjidhada thyroid-ka ee isticmaalka iodine si loo soo saaro hoormoonka tayroodh. Waxa kale oo ay xakameysaa beddelaadda hoormoonka thyroid T4 ee T3. PTU waxay leedahay waqti gaaban, sidaas darteed bukaanada qaadanaya dawadan sida caadiga ah waxaa lagu faray in ay qaataan daawada laba illaa seddex jeer maalintii si loo yareeyo heerarka hoormoonka tayroodh.
PTU waxay leedahay saameyno badan oo ka yimaada daawooyinka kale ee halkan looga wada hadlay, waana daawada loo doorbidayo hyperthyroidism kaliya xaaladaha yar (inta lagu jiro xilliga hore ee uurka, duufaanka aadka u daran iyo marka uu bukaanku la kulmo dhibaatooyin culus oo ka yimaada methimazole).
Dalka Mareykanka, kaliya PTU waa la heli karaa; ma jiro magac calaamad ah oo PTU ah oo laga iibsaday Maraykanka. Qaar ka mid ah shirkadaha wax soo saarka ayaa soo saaraan PTU.
Macluumaad Dheeraad ah
Wax badan ka ogow hyperthyroidism iyo daaweyntiisa, oo ay ku jiraan daawooyinka antithyroid, khayraadkan:
- Hyperthyroidism | Jirro 'Cudurrada' Qanjirka 'Overactive'
- Jirrada 'Cudurrada' iyo Hyperthyroidism 101
- Khatarta Cudurrada / Calaamadaha Helitaanka Hyperthyroidism
- Khatarta Cudurka Dhiigga iyo Hyperthyroidism
- Su'aalaha Inta Badan La Isweydiiyo ee ku Saabsan Cudurka Hyperthyroidism iyo Cudurka Qallalka
- 3 Waddooyinka lagu daaweeyo Hyperthyroidism
Ilaha:
Daily Med, Daawooyinka Daawooyinka Cunnada iyo Dawooyinka Cunnada Maraykanka, Online
Isgaarsiinta Badbaadinta Daroogada ee FDA: Digniinta Cusub ee Cusub ee ku saabsan dhaawaca beerka ee ba'an ee propylthiouracil, Abriil 21, 2010, Online
Ross, Douglas MD, "Macluumaadka bukaanka: Daawooyinka Antithyroid," UpToDate . Last updated: November 13, 2009