Prezcobix (darunavir + cobicistat) waa daawo loo isticmaalo daawada antiretroviral oo loo isticmaalo daaweynta HIV . Labada qaybood ee daroogada ku jira ee Prezcobix ayaa si shakhsiyan ah loo iibsadaa ka hor intaan la helin qiimaha la yiraahdo Prezista (darunavir) iyo Tybost (cobicistat) .
Kiniinka kelida ah, kiniin la isku qaabeeyey ayaa si fudud u bixiya, qiyaasta daawada maalinlaha ah, iyada oo qayb ka mid ah geedi-socodka loo yaqaan 'cobicistat' si waxtar leh u kordha iyo joogtaynta qadarka plasma ee qiyaasta jirka ee jirka.
Prezcobix waxaa ansixiyay Maamulka Cunnada iyo Mukhaadaraadka ee Maraykanka (FDA) bishii Janaayo 2015 ee loogu talagalay bukaanada qaangaarka ah ee qibrada leh ee cusub ee qaba HIV-1.
Foomka
Kiniiniga xayawaanka ah ee la duubay, oo ka kooban 800mg oo ah darunavir iyo 150mg of cobicistat, waa midab casaan ah oo ku daboolay "TG" hal dhinac iyo "800" oo kale.
Qiyaasta
Hal kiniin ayaa maalin walba la qaataa cunto. Prezcobix looma isticmaali karo kali ah, lakiin waa in la qaato si wadajir ah hal ama dhowr daawo oo daawooyinka loo yaqaan 'antiretroviral drugs'.
Tilmaamaha
Ka hor inta aan la bilaabin, bukaanku waa in la baaraa si loo qiimeeyo qiyaasta loo yaqaan 'cynineine' ee lagu qiyaasay maaddaama uu Prezcobix uu awood u yeelan karo inuu kiciyo shaqada kelyaha (kelyaha), badanaaba bukaanka qaba cillad aan hagaagsanayn ama aan la ogaan karin. Markii lagala wareegay Viread (Tenofovir) - daroogada ayaa sidoo kale loo yaqaan in ay keento xayawaanka xayawaanka ee qaar ka mid ah-waxaa lagu talinayaa in bukaanku la baadho qiyaasta nadiifinta, dhalashada kaadida, iyo borotiin kaadida.
Waxaa sidoo kale lagu talinayaa in bukaanada daaweyn-khibrad leh, gaar ahaan kuwa ku faafay xannuunka HIV protease , la siiyo baaritaanka iska caabinida hiddaha ka hor intaysan qaadin Prezcobix. Haddii baaritaanka unugyada aan la helin, waa in laga fogaadaa konkobixiska loogu talagalay qof kasta oo horey u soo gaadhay xannibaadaha HIV ee protease.
Saameynada Caadiga ah
Qaybta 3aad ee cilmi-baarista bani'aadamka ee bani'aadamnimada, tiro badan oo saameyn ku yeelashada daroogada ayaa la ogaaday markii la isticmaalayo Prezcobix. Dhacdooyinka ugu caansan, ee lagu soo sheegay 5% ama ka yar bukaanada, waxay ahaayeen:
- Shuban
- Lalabbo
- Finan
- Madax xanuun
- Calool xanuun
- Matagid
Astaamaynta Daroogada
Prezcobix waa in aan lagu qaadin daawooyinka soo socda ama daawooyinka dabiiciga ah:
- Daawada anti-anginal: Ranexa
- Daawooyinka isdaba joogga ah: Multaq
- Dawooyinka anti-cholesterol: Mevacor, Zocor
- Dawooyinka lidka ku ah daawooyinka: Uroxatral
- Dawooyinka anti-hypertension: Revatio
- Daawooyinka ka hortagga maskaxda: Latuda, Orap
- Dawooyinka Kansarka: Camptosar, Campto
- Ergot-ka kooban walxaha dheef-shiid kiimiko ah: DHE 45, Ergotrate, Hydergine, Migranal
- Dawooyinka anti-tuberculosis ku salaysan Rifampin: Mycobutin, Rifater, Rifamate, Rimactane, Rifadin, Priftin
- Sedatives: Dormicum, Halcion, Hypam, Hyponvel, Trilam, Aasaasay
- St. John Wort
Isdhex galka daawada Antiretroviral
Isticmaalka konkobixix daroogada daawooyinka antiretrovoviral ayaa laga yaabaa in ay keenaan in lumiyo saameynta daaweynta ee daroogada raacsan ama khatarta sii kordheysa ee saameynaha kale:
- Crixivan (indinavir) looma ogolaanayo in lagu soo celiyo degmada Prezcobix.
- Videox (didanosine) waa in la qaataa hal saac ka hor ama hal saac ka dib qaadashada koncobix.
- Intel'ka (etravirine) waa in aan lagu xirin koncobix.
- Viramune (nevirapine) waa in aan lagu sii deynin degmada Prezcobix
- Selzentry (maraviroc) qiyaasta waa in la isku hagaajiyaa ilaa 150mg laba goor maalintii, haddii lagu sii daayo Prezcobix.
Isdhexgalka kale ama Tixgelinnada kale
- U sheeg dhakhtarkaaga wixii xaalad ah ee kalyaha ama kalyaha ah ee la og yahay ama laga shakiyay (kelyo) laga yaabo inaad horey u soo qaadatay ka hor.
- Daawada maqnaashaha aan habooneyn (Viagra, Levitra, Cialis) waa in loo adeegsadaa taxadar leh maaddaama ay ka mid tahay qaybta rugicistat ee kudhisan Koncobix waxay kor u qaadi kartaa heerarka saameynta liddiga ah, oo ay ku jiraan waxyeelo muuqda, isku-buuqsanaanta, iyo horjoogsiga (xannuuno xanuun, joogsi joogta ah). Waxaa lagu talinayaa in Viagra qiyaasta hoos loo dhigo in ka badan 25mg 48 saacadood; Qiyaasta Levitra waa la yareeyey in ka badan 2.5mg 72 saacadood, iyo qiyaasta Cialis waa la yareeyey in ka badan 10mg 72 saacadood.
Ilaha:
Bristol-Myers Squibb. "PREZCOBIX - MACLUUMAAD KU QORAN MACLUUMAAD". New York, New York